... plasticity mechanisms were unrecognized, and have important implications for the therapeutic use of cannabinoid receptor antagonists in humans,” concluded Bear and colleagues.
Citing the development ...
... antagonist CP 96,345, but not the glucocorticoid receptor antagonist RU486, increased NK cell activity. ... role of serotonergic agents and substance P antagonists in improving natural killer cell innate ...
... and thereby blood pressure. He added that some patients may also benefit from adding mineralocorticoid receptor antagonists (MRAs) to their treatment regimens. MRAs have traditionally been used to ...
... to move forward with a phase 1 clinical trial using this FDA-approved GRP receptor antagonist for neuroblastoma," Chung said. "We hope to demonstrate the safety of targeting GRP receptors for ...
... the brain. Unpublished findings from our laboratory suggest that, similar to MK-571, other leukotriene receptor antagonists, e.g. montelukast (SingulairTM) and zafirlukast (AccolateTM) can suppress ...
... these interesting research findings in animals with the lack of antidepressant efficacy of a CRF1 receptor antagonist in the Pfizer study? Is this approach simply ineffective in humans or might ...
... is the treatment of choice. When medical therapy is needed, the guideline recommends patients be treated with mineralocorticoid receptor antagonists, drugs which inhibit the action of aldosterone.
... first of a new class of HIV drugs called CCR5 receptor antagonists, has been shown to be effective over 48 weeks for drug-resistant patients with R5 HIV-1, a variation of ...
... of esophagitis). In these uses, proton pump inhibitors (PPIs) are more effective than histamine receptor antagonists (H2RAs), which are more effective than placebo. II. Long-term use of PPIs for ...
... Connecticut Healthcare System, comments: "The NMDA receptor antagonist model and the EAAT1 knockout animal ... ago, such as the group II metabotropic glutamate receptor agonists."
Dr. Holmes does note ...
... of their consumed food and are resistant to diet-induced obesity. Also, small-molecule ghrelin receptor antagonists have been shown to reduce food intake, promote selective weight loss in the form of ...
... that many of the hypnotic medications that are most effective in treating insomnia are benzodiazepine receptor antagonists (BzRAs), which increase activity at the GABA neurons. According to a new ...
... a gene in the affected joint, he was able to stimulate production of a human interleukin-1 receptor antagonist protein, which serves to block actions of the interleukin-1 protein.
"The idea is that ...
... proton pump inhibitor pantoprazole or with other acid-lowering medications called H2 receptor antagonists.
Previous research indicates that proton pump inhibitors other than pantoprazole can block ...
... for rheumatoid arthritist include anakinra (Kineret®, an IL-1 receptor antagonist) and etanercept (Enbrel®, a tumor necrosis factor blocker)," said Farshid Guilak, Ph.D., study scientist ...